LIGAND-GATED ION CHANNEL SUBUNITS

Voltage-gated ion channel subunits |  Download ion channel data as an Excel file

5-HT3 receptors
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
5-HT3 receptors 5-hydroxytryptamine 5-HT3A HTR3A Htr3a Htr3a
5-HT3 receptors 5-hydroxytryptamine 5-HT3B HTR3B Htr3b Htr3b
5-HT3 receptors 5-hydroxytryptamine 5-HT3C HTR3C
5-HT3 receptors 5-hydroxytryptamine 5-HT3D HTR3D
5-HT3 receptors 5-hydroxytryptamine 5-HT3E HTR3E
5-HT3 receptors 5-hydroxytryptamine 5-HT3AB
5-HT3 receptors 5-hydroxytryptamine 5-HT3A
GABAA receptors
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
GABAA receptors GABA α1 GABRA1 Gabra1 Gabra1
GABAA receptors GABA α2 GABRA2 Gabra2 Gabra2
GABAA receptors GABA α3 GABRA3 Gabra3 Gabra3
GABAA receptors GABA α4 GABRA4 Gabra4 Gabra4
GABAA receptors GABA α5 GABRA5 Gabra5 Gabra5
GABAA receptors GABA α6 GABRA6 Gabra6 Gabra6
GABAA receptors GABA β1 GABRB1 Gabrb1 Gabrb1
GABAA receptors GABA β2 GABRB2 Gabrb2 Gabrb2
GABAA receptors GABA β3 GABRB3 Gabrb3 Gabrb3
GABAA receptors GABA γ1 GABRG1 Gabrg1 Gabrg1
GABAA receptors GABA γ2 GABRG2 Gabrg2 Gabrg2
GABAA receptors GABA γ3 GABRG3 Gabrg3 Gabrg3
GABAA receptors GABA δ GABRD Gabrd Gabrd
GABAA receptors GABA ε GABRE Gabre Gabre
GABAA receptors GABA θ GABRQ Gabrq Gabrq
GABAA receptors GABA π GABRP Gabrp Gabrp
GABAA receptors GABA ρ1 GABRR1 Gabrr1 Gabrr1
GABAA receptors GABA ρ2 GABRR2 Gabrr2 Gabrr2
GABAA receptors GABA ρ3 GABRR3 Gabrr3 Gabrr3
Glycine receptors
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
Glycine receptors glycine α1 GLRA1 Glra1 Glra1
Glycine receptors glycine α2 GLRA2 Glra2 Glra2
Glycine receptors glycine α3 GLRA3 Glra3 Glra3
Glycine receptors glycine α4 (pseudogene in humans) GLRA4 Glra4 Glra4
Glycine receptors glycine β GLRB Glrb Glrb
Glycine receptors glycine Glycine Receptor (All subtypes)
Nicotinic acetylcholine receptors
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
Nicotinic acetylcholine receptors acetylcholine α1 CHRNA1 Chrna1 Chrna1
Nicotinic acetylcholine receptors acetylcholine α2 CHRNA2 Chrna2 Chrna2
Nicotinic acetylcholine receptors acetylcholine α3 CHRNA3 Chrna3 Chrna3
Nicotinic acetylcholine receptors acetylcholine α4 CHRNA4 Chrna4 Chrna4
Nicotinic acetylcholine receptors acetylcholine α5 CHRNA5 Chrna5 Chrna5
Nicotinic acetylcholine receptors acetylcholine α6 CHRNA6 Chrna6 Chrna6
Nicotinic acetylcholine receptors acetylcholine α7 CHRNA7 Chrna7 Chrna7
Nicotinic acetylcholine receptors acetylcholine α9 CHRNA9 Chrna9 Chrna9
Nicotinic acetylcholine receptors acetylcholine α10 CHRNA10 Chrna10 Chrna10
Nicotinic acetylcholine receptors acetylcholine β1 CHRNB1 Chrnb1 Chrnb1
Nicotinic acetylcholine receptors acetylcholine β2 CHRNB2 Chrnb2 Chrnb2
Nicotinic acetylcholine receptors acetylcholine β3 CHRNB3 Chrnb3 Chrnb3
Nicotinic acetylcholine receptors acetylcholine β4 CHRNB4 Chrnb4 Chrnb4
Nicotinic acetylcholine receptors acetylcholine γ CHRNG Chrng Chrng
Nicotinic acetylcholine receptors acetylcholine δ CHRND Chrnd Chrnd
Nicotinic acetylcholine receptors acetylcholine ε CHRNE Chrne Chrne
P2X receptors
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
P2X receptors ATP P2X1 P2RX1 P2rx1 P2rx1
P2X receptors ATP P2X2 P2RX2 P2rx2 P2rx2
P2X receptors ATP P2X3 P2RX3 P2rx3 P2rx3
P2X receptors ATP P2X4 P2RX4 P2rx4 P2rx4
P2X receptors ATP P2X5 P2RX5 P2rx5 P2rx5
P2X receptors ATP P2X6 P2RX6 P2rx6 P2rx6
P2X receptors ATP P2X7 P2RX7 P2rx7 P2rx7
ZAC
Family name Ligand Official IUPHAR receptor name Human gene name Rat gene name Mouse gene name Comment
ZAC Zn++ ZAC ZACN

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